About 5 results found for searched term "CGRP antagonist 1" (0.49 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M50213 | CGRP antagonist 1 | CGRP Receptor |
| CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki and IC50 values of 1.7 nM and 5.7 nM, respectively. | ||
| M2133 | MK-3207 hydrochloride | CGRP Receptor |
| MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM. | ||
| M3618 | MK-0974 | CGRP Receptor |
| Telcagepant | ||
| MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively. | ||
| M10372 | Vazegepant hydrochloride | CGRP Receptor |
| Zavegepant, BHV-3500 hydrochloride | ||
| Vazegepant (BHV-3500) hydrochloride is a first-in-class, high affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM). Vazegepant hydrochloride may be useful in the effective treatment of lung inflammation associated with COVID-19. | ||
| M13933 | MK-3207 | CGRP Receptor |
| MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3. | ||
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